compound
stringlengths
4
309
solvents
stringclasses
27 values
gradient
stringclasses
57 values
column
stringclasses
34 values
flow_rate
float64
0.01
3
temp
float64
25
65
rt
float64
0
6.03k
source
stringclasses
8 values
method_number
int64
1
73
Br.Br.CC=1C=CN=C(CN)C1O
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
13.806
enaminert
2
Br.Br.NC1(CC1)C2=CSC=N2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
8.856
enaminert
2
Br.BrC1=NC=2CCNCCC2S1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
34.734
enaminert
2
Br.BrC=1C=CC=C(C1)C2=CSC(=N2)C3=CC=CO3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
93.378
enaminert
2
Br.BrC=1C=CC=CC1C2=CSC(NC=3C=CC=CN3)=N2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
76.716
enaminert
2
Br.CC(=O)NC1(C)CNC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
9.834
enaminert
2
Br.CC1=NN=C2SC(N)=NN12
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
15.072
enaminert
2
Br.CC1CNCCC=2C=CC(O)=CC12
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
20.862
enaminert
2
Br.CC=1C=CC(=O)NC1N
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
25.596
enaminert
2
Br.CCC(C)C1=CSC(N)=N1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
39.762
enaminert
2
Br.CCCNC(=NCCNC(=O)C=1C=CC(Br)=CC1)N
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
57.204
enaminert
2
Br.CN1CCC1CBr
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
10.308
enaminert
2
Br.ClC=1C=NC=CC1C(=O)CBr
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
67.242
enaminert
2
Br.OC(=O)C1(CCCN1)C(F)(F)F
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
11.088
enaminert
2
Br.OC(=O)C1=CSC=2C(Br)=CC=NC12
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
57.756
enaminert
2
BrC(=CC=1C=CC=CC1)C=NNC(=O)C2=CC(=NN2)C3CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
72.804
enaminert
2
BrC1(Br)CC(C1)C(=O)OCCOCC=2C=CC=CC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
80.04
enaminert
2
BrC1=C(N=C2CCCN12)C(=O)NC(C3CCCC3)C(=O)N4CCN5CCOCC5C4
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
45.504
enaminert
2
BrC1=CC(I)=CNC1=O
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
58.812
enaminert
2
BrC1=CC=C(CNC2(CC=C)CCOC2)S1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
30.78
enaminert
2
BrC1=CC=C(O1)C(=O)NNC(=S)NCC=2C=CC=CC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
65.718
enaminert
2
BrC1=CC=C(O1)C2=NN=C(CN3CCCCC3C4=NC=5C=CC=CC5S4)O2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
89.898
enaminert
2
BrC1=CC=C(S1)C(=O)COC(=O)CCC2=CNC=3C=CC=CC23
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
84.204
enaminert
2
BrC1=CC=C(S1)C2(CNCC=3C=CNN3)CCC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
57.612
enaminert
2
BrC1=CC=C(S1)C2=CSC(NC(=O)C=3C=NC=CN3)=N2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
82.776
enaminert
2
BrC1=CC=C(S1)C2=NOC(=N2)C3CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
47.508
enaminert
2
BrC1=CC=C(S1)S(=O)(=O)NC(=O)C=2C=NC=3SC=CC3C2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
63.006
enaminert
2
BrC1=CC=C(S1)S(=O)(=O)NC(=O)CC2OCCC=3SC=CC23
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
69
enaminert
2
BrC1=CC=C(S1)S(=O)(=O)NC=2C=CC(=CC2)C(=O)NCCC=3C=CC=CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
78.258
enaminert
2
BrC1=CN(CC(=O)NC=2C=CN=C(SC=3C=CC=CN3)C2)C(=O)NC1=O
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
47.328
enaminert
2
BrC1=CN(CCNCC2CC32CCCCC3)N=N1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
39.876
enaminert
2
BrC1=CN=C2C(NCCC3CCC(=O)N3)=NC=NN12
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
55.29
enaminert
2
BrC1=CNC(=O)C=2C=CC=NC12
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
44.808
enaminert
2
BrC1=CNC=2C=C(C=NC12)C3=NC(CN4C=CN=N4)=NO3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
47.826
enaminert
2
BrC1=CSC(=C1)C2=NN=C3CCOCCN23
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
63.846
enaminert
2
BrC1=CSC(=C1)C2=NN=C3N2CCCC43CCOCC4
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
62.832
enaminert
2
BrC1=CSC(CN2N=C3COCCN3C2=O)=C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
65.892
enaminert
2
BrC1=CSC(CNC(=O)N2CCOCC2)=C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
55.896
enaminert
2
BrC1=CSC=C1CNC=2C=CC(=O)NN2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
50.544
enaminert
2
BrC1=CSN=C1OCC2=NC(C#N)=CS2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
79.824
enaminert
2
BrC1=NOC(C2CC2)=C1C(=O)OCC3=CC=4C=CC=CC4NC3=O
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
43.134
enaminert
2
BrC1=NSC(=N1)N(CCOC2CC2)CC=3C=CSC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
79.038
enaminert
2
BrC1=NSC=C1C(=O)N[C@H]2C[C@@H](C2)C3=NN=C4CCCCCN34
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
53.85
enaminert
2
BrC=1C(NCC2=NN=C(O2)C3CCC3)=CC=C4SC=NC14
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
72.846
enaminert
2
BrC=1C=C(C#N)C2=NC=NN2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
54.306
enaminert
2
BrC=1C=C(C#N)C=C(C1)N2C=C(N=N2)C3COCCO3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
71.91
enaminert
2
BrC=1C=C(C=CC1C#N)N2CCC(CC2)C3=NC=CO3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
82.806
enaminert
2
BrC=1C=C(C=O)C2=NNC=C2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
69.804
enaminert
2
BrC=1C=C(CC2=NOC(=N2)[C@@H]3C[C@H]4CC[C@@H]3O4)C=C5OCCOC15
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
78.99
enaminert
2
BrC=1C=C(CN(CC2=NOC=3CCCCC23)S(=O)(=O)C=C)C=C4OCCOC14
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
88.74
enaminert
2
BrC=1C=C(CN2C(=O)[C@H]3CCCN3S2(=O)=O)C=CN1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
71.496
enaminert
2
BrC=1C=C(CN2C=C(N=N2)C=3C=NN(CC(=O)NC(C4CC4)C5=NC=CS5)C3)NN1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
65.628
enaminert
2
BrC=1C=C(CNC2=CN(CC=3C=CC=CC3)N=N2)C=CN1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
72.216
enaminert
2
BrC=1C=C(NC(=O)CCN2CCOCC2)C=CC1C#C
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
41.652
enaminert
2
BrC=1C=C(NC=2C=C3COCCN3N2)N=CN1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
54.918
enaminert
2
BrC=1C=C(NCC=2C=CON2)C=C3OCCCOC13
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
76.278
enaminert
2
BrC=1C=C2N=CC=CC2=CC1OC=3N=NC=4CCCC4C3C#N
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
78.756
enaminert
2
BrC=1C=C2NN=CC2=NC1Br
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
68.016
enaminert
2
BrC=1C=CC(=C(C#N)C1)N2C=CN=N2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
62.568
enaminert
2
BrC=1C=CC(=CC1)C(=O)CSC2=NN=NN2C=3C=CC=CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
84.486
enaminert
2
BrC=1C=CC(=CC1)C(=O)NC2=CC(=NN2)C3CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
67.032
enaminert
2
BrC=1C=CC(=CC1)C(=O)NCCC(=O)NC=2C=CC=NC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
52.518
enaminert
2
BrC=1C=CC(=CC1)C(=O)NCCC(=O)NCC2(CCCCC2)N3CCOCC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
49.626
enaminert
2
BrC=1C=CC(=CC1)C2(CC2)NS(=O)(=O)CC=3C=CC=CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
80.28
enaminert
2
BrC=1C=CC(=CC1)C2=NNC(CNC(=O)C=3C=CC=C4C(=O)NN=CC34)=N2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
63.282
enaminert
2
BrC=1C=CC(=CC1)C2CCCN2C(=O)C#C
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
67.71
enaminert
2
BrC=1C=CC(=CC1)C=2C=CN=C(N2)N3CCC(C3)N4CC=CC4
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
91.692
enaminert
2
BrC=1C=CC(=CC1)C=2N=NN(CC3=CC(=O)N4C=CSC4=N3)N2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
65.454
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)CC2COC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
60.102
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)CCN2N=NC(=N2)C=3C=CC=CC3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
77.94
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)N2CCCCC2C(=O)NNC(=O)C=3C=CC=CN3
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
71.646
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)N2CCN(CC3=CC(=O)N4C(=CSC4=N3)C=5C=CC=CC5)CC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
68.994
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)NC2CCC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
80.37
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)NC=2C=CC=C3C=CC=NC23
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
85.62
enaminert
2
BrC=1C=CC(=CC1)S(=O)(=O)NCC=2C=CC(CN3C=CN=C3)=CC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
55.11
enaminert
2
BrC=1C=CC(=CC1)[C@H]2C[C@@H](C2)NC(=O)NC3CCCC3C#N
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
76.638
enaminert
2
BrC=1C=CC(=CC1C(=O)NC=2C=CC=C3C=CC=CC23)S(=O)(=O)N4CCCC4
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
81.684
enaminert
2
BrC=1C=CC(=NN1)N2CCOCC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
55.722
enaminert
2
BrC=1C=CC(=O)N(CC(=O)N2CCC3(C2)CCCOC3)C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
56.082
enaminert
2
BrC=1C=CC(C#N)=NC1N2CCN(CC=3N=CNN3)CC2
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
49.032
enaminert
2
BrC=1C=CC(CN(CC=C)C=2N=CN=C(N2)N3CCOCC3)=CC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
92.772
enaminert
2
BrC=1C=CC(CN2C=C(N=N2)C=3C=NC=NC3)=CC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
74.376
enaminert
2
BrC=1C=CC(CN2CCN(CC2)C(=O)C3=CC=C(S3)C4=CC=CO4)=NC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
65.058
enaminert
2
BrC=1C=CC(NCC2=NN=C(O2)C3CC3)=C4CCCCC14
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
85.962
enaminert
2
BrC=1C=CC(NS(=O)(=O)C=2C=CC=CC2)=CC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
76.566
enaminert
2
BrC=1C=CC(OC=2C=CC=C(NC(=O)C=3C=CC=C(C#CC4CC4)C3)C2)=CC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
94.668
enaminert
2
BrC=1C=CC(OCC2=NC(CN3C=CC=CC3=O)=NO2)=CN1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
52.26
enaminert
2
BrC=1C=CC(SCC#N)=CC1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
74.16
enaminert
2
BrC=1C=CC2=NC=3CCNCC3N2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
16.734
enaminert
2
BrC=1C=CC2=NC=CC(=O)N2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
54.576
enaminert
2
BrC=1C=CC=2C(=NN=CC2C1)N3CC[C@@H](C3)OC4CC4
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
46.59
enaminert
2
BrC=1C=CC=2C(=O)C(=O)C=3C=CC=CC3C2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
84.468
enaminert
2
BrC=1C=CC=2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
57.942
enaminert
2
BrC=1C=CC=2C(=O)N(CCC(=O)NC=3C=CC=NC3)C(=O)C2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
53.676
enaminert
2
BrC=1C=CC=2C=C(NC2C1)C(=O)NCC(N3CCOCC3)C4=CC=CS4
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
62.634
enaminert
2
BrC=1C=CC=2C=NC=CC2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
37.866
enaminert
2
BrC=1C=CC=2N=C(CN3CCCC(C3)C=4C=CC=CC4)NC(=O)C2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
69.12
enaminert
2
BrC=1C=CC=2N=CN(CCN3C=CC=N3)C(=O)C2N1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
44.826
enaminert
2
BrC=1C=CC=2NC(=O)COC2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
66.498
enaminert
2
BrC=1C=CC=2NC(=S)OC2C1
{'A': [{'CC#N': 95, 'O': 5}, {'C(=O)O': 0.0265}], 'B': [{'O': 100}, {'C(=O)O': 0.0265}]}
[(0, 99), (0.01, 99), (1.5, 0), (1.73, 0), (1.74, 99), (2, 99)]
('RP', 4.6, 30, 2.7)
3
30
55.302
enaminert
2